Jon Clardy, PhD
Hsien Wu and Daisy Yen Wu Professor of Biological Chemistry and Molecular Pharmacology, Harvard Medical School
Protein evolution: when two become three.
Identification and validation of tetracyclic benzothiazepines as Plasmodium falciparum cytochrome bc1 inhibitors.
Authors: Authors: Dong CK, Urgaonkar S, Cortese JF, Gamo FJ, Garcia-Bustos JF, Lafuente MJ, Patel V, Ross L, Coleman BI, Derbyshire ER, Clish CB, Serrano AE, Cromwell M, Barker RH, Dvorin JD, Duraisingh MT, Wirth DF, Clardy J, Mazitschek R.
Chem Biol
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Chem Biol
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Sceliphrolactam, a polyene macrocyclic lactam from a wasp-associated Streptomyces sp.
A non-radioactive DAPI-based high-throughput in vitro assay to assess Plasmodium falciparum responsiveness to antimalarials--increased sensitivity of P. falciparum to chloroquine in Senegal.
Authors: Authors: Ndiaye D, Patel V, Demas A, LeRoux M, Ndir O, Mboup S, Clardy J, Lakshmanan V, Daily JP, Wirth DF.
Am J Trop Med Hyg
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Am J Trop Med Hyg
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Identification and characterization of small molecule inhibitors of a class I histone deacetylase from Plasmodium falciparum.
Authors: Authors: Patel V, Mazitschek R, Coleman B, Nguyen C, Urgaonkar S, Cortese J, Barker RH, Greenberg E, Tang W, Bradner JE, Schreiber SL, Duraisingh MT, Wirth DF, Clardy J.
J Med Chem
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J Med Chem
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Codinaeopsin, an antimalarial fungal polyketide.
High-throughput Plasmodium falciparum growth assay for malaria drug discovery.
Authors: Authors: Baniecki ML, Wirth DF, Clardy J.
Antimicrob Agents Chemother
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Antimicrob Agents Chemother
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Total synthesis of psammaplysenes A and B, naturally occurring inhibitors of FOXO1a nuclear export.
The biosynthetic gene cluster of Pantocin a provides insights into biosynthesis and a tool for screening.
Authors: Authors: Jin M, Wright SA, Beer SV, Clardy J.
Angew Chem Int Ed Engl
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Angew Chem Int Ed Engl
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Synthesis and biological evaluation of analogues of the antibiotic pantocin B.