Obesity is a growing worldwide health epidemic that is placing ever-growing medical and economic burdens on society. The prevalence of the associated condition non-alcoholic fatty liver disease (NAFLD) is also rising, and this condition is now the leading cause of chronic liver disease in the West. As a result of the multifaceted nature of these diseases and the lack of mechanistic understanding of their molecular underpinnings, doctors must resort to “trial and error” to identify effective treatments. The goal of this research is to develop small molecules that modulate gut bacterial metabolism of bile acids, compounds that play crucial roles in human metabolism, as new potential treatments for metabolic syndrome and NAFLD. These first-in-class molecules that target the microbiota will also allow us to better understand how the human microbiome contributes to obesity on a molecular level, knowledge that will pave the way for the development of future microbiome-based therapies.

Funding

Funding Duration

July 1, 2018 - June 30, 2019

Funding level

Pilot

People

Principal Investigator

Sloan Devlin

PhD
Associate Professor of Biological Chemistry and Molecular Pharmacology, Harvard Medical School
Co-PI

Arijit Adhikari

PhD
Research Fellow in Biological Chemistry and Molecular Pharmacology (INT), Harvard Medical School

Intellectual Property

Publications

Patents

WO2020231776
:
Small molecule modulators of gut bacterial bile acid metabolism
(Patent application)